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ABCG2 gene
Gene • C1332002
Definition
This gene plays a role in xenobiotic transport and multi-drug resistance.
Synonyms
ABCG2 gene • BREAST CANCER RESISTANCE PROTEIN • ATP-Binding Cassette, Sub-Family G (WHITE), Member 2 Gene • ABCG2 • ABCP • ATP-BINDING CASSETTE TRANSPORTER, PLACENTA-SPECIFIC • BCRP • EST157481 • MITOXANTRONE-RESISTANCE PROTEIN • MRX • MXR • ATP-binding cassette, sub-family G (WHITE), member 2 • ATP-BINDING CASSETTE, SUBFAMILY G, MEMBER 2 • CD338
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Protein Binding
integral to membrane
Cyclosporine
Cell membrane
7,8-Dihydro-7,8-dihydroxybenzo(a)pyrene 9,10-oxide
Benzo(a)pyrene
Tetrachlorodibenzodioxin
ATP binding
nucleotide binding
Estradiol
arsenic trioxide
Aflatoxin B1
pirinixic acid
Tretinoin
Fluorouracil
decitabine
Progesterone
Biological Transport
sodium arsenite
Transmembrane Transport
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Related concepts
#
|
Concept name
|
Type
|
Relation
|
Support
|
Score
|
1
|
ABCB1 gene
|
Gene
|
Inferred
|
Explain
|
0.30646
|
2
|
GF 120918
|
Compound
|
Known
|
Explain
|
0.28992
|
3
|
MIR520H gene
|
Gene
|
Known
|
Explain
|
0.28510
|
4
|
taxane
|
Compound
|
Known
|
Explain
|
0.26762
|
5
|
2-pyrrolino-DOX
|
Compound
|
Known
|
Explain
|
0.26762
|
6
|
tectochrysin
|
Compound
|
Known
|
Explain
|
0.26762
|
7
|
6-prenylchrysin
|
Compound
|
Known
|
Explain
|
0.26762
|
8
|
albendazole sulfoxide
|
Compound
|
Known
|
Explain
|
0.26511
|
9
|
oxfendazole
|
Compound
|
Known
|
Explain
|
0.26511
|
10
|
AN 215
|
Compound
|
Known
|
Explain
|
0.23183
|
11
|
2-pyrrolino-DOX-14-O-glt-RC-121
|
Compound
|
Known
|
Explain
|
0.21781
|
12
|
6-bromoindirubin-3'-oxime
|
Compound
|
Known
|
Explain
|
0.21651
|
13
|
Flavones
|
Compound
|
Known
|
Explain
|
0.21413
|
14
|
SDZ PSC 833
|
Compound
|
Known
|
Explain
|
0.19836
|
15
|
pantoprazole
|
Compound
|
Known
|
Explain
|
0.19742
|
16
|
dibenzoylmethane
|
Compound
|
Known
|
Explain
|
0.19453
|
17
|
xenobiotic-transporting ATPase activity
|
Function
|
Known
|
Explain
|
0.19411
|
18
|
bis((3R,5S,6E)-7-(2-cyclopropyl-4-(4-fluorophenyl)-3-quinolyl)-3,5-dihydroxy-6-heptenoate), monocalcium salt
|
Compound
|
Known
|
Explain
|
0.18804
|
19
|
Cyclosporins
|
Compound
|
Known
|
Explain
|
0.18777
|
20
|
Digoxin
|
Compound
|
Known
|
Explain
|
0.17912
|
21
|
Bay w 6228
|
Compound
|
Known
|
Explain
|
0.17010
|
22
|
estrone sulfate
|
Compound
|
Known
|
Explain
|
0.16333
|
23
|
Triamcinolone
|
Compound
|
Known
|
Explain
|
0.16266
|
24
|
benzo(k)fluoranthene
|
Compound
|
Known
|
Explain
|
0.15877
|
25
|
flavone
|
Compound
|
Known
|
Explain
|
0.14963
|
26
|
artesunate
|
Compound
|
Known
|
Explain
|
0.14840
|
27
|
MIR328 gene
|
Gene
|
Known
|
Explain
|
0.14832
|
28
|
ABCC1 gene
|
Gene
|
Inferred
|
Explain
|
0.14410
|
29
|
heme transporter activity
|
Function
|
Known
|
Explain
|
0.14153
|
30
|
2-amino-1-methyl-6-phenylimidazo(4,5-b)pyridine
|
Compound
|
Known
|
Explain
|
0.14068
|
31
|
AG 1343
|
Compound
|
Known
|
Explain
|
0.13419
|
32
|
Pravastatin
|
Compound
|
Known
|
Explain
|
0.13326
|
33
|
Methylprednisolone
|
Compound
|
Known
|
Explain
|
0.13216
|
34
|
heme transport
|
Function
|
Known
|
Explain
|
0.13178
|
35
|
oltipraz
|
Compound
|
Known
|
Explain
|
0.12725
|
36
|
2-tert-butylhydroquinone
|
Compound
|
Known
|
Explain
|
0.12583
|
37
|
Beclomethasone
|
Compound
|
Known
|
Explain
|
0.12081
|
38
|
Epirubicin
|
Compound
|
Known
|
Explain
|
0.11498
|
39
|
Rokan
|
Compound
|
Known
|
Explain
|
0.10299
|
40
|
Omeprazole
|
Compound
|
Known
|
Explain
|
0.09791
|
41
|
Silymarin
|
Compound
|
Known
|
Explain
|
0.09776
|
42
|
Corticosterone
|
Compound
|
Known
|
Explain
|
0.09773
|
43
|
Anticonvulsants
|
Compound
|
Known
|
Explain
|
0.09720
|
44
|
ABC-2 type transporter
|
Domain
|
Known
|
Explain
|
0.09585
|
45
|
Depsipeptides
|
Compound
|
Known
|
Explain
|
0.09470
|
46
|
urate metabolic process
|
Function
|
Known
|
Explain
|
0.08877
|
47
|
Cimetidine
|
Compound
|
Known
|
Explain
|
0.08839
|
48
|
indolo(3,2-b)carbazole
|
Compound
|
Known
|
Explain
|
0.08639
|
49
|
Nitrofurantoin
|
Compound
|
Known
|
Explain
|
0.07238
|
50
|
monoisoamyl-2,3-dimercaptosuccinate
|
Compound
|
Known
|
Explain
|
0.07159
|
51
|
Luteolin
|
Compound
|
Known
|
Explain
|
0.06513
|
52
|
chrysin
|
Compound
|
Known
|
Explain
|
0.06393
|
53
|
ABCB4 gene
|
Gene
|
Inferred
|
Explain
|
0.06112
|
54
|
indole-3-carbinol
|
Compound
|
Known
|
Explain
|
0.05910
|
55
|
20-Methylcholanthrene
|
Compound
|
Known
|
Explain
|
0.05890
|
56
|
ABC transporters - Homo sapiens (human)
|
Pathway
|
Known
|
Explain
|
0.05758
|
57
|
Rifampin
|
Compound
|
Known
|
Explain
|
0.04959
|
58
|
CS 045
|
Compound
|
Known
|
Explain
|
0.04876
|
59
|
ZD1839
|
Compound
|
Known
|
Explain
|
0.04503
|
60
|
PIM1 gene
|
Gene
|
Known
|
Explain
|
0.04227
|
61
|
Phenobarbital
|
Compound
|
Known
|
Explain
|
0.04126
|
62
|
KEGG:hsa04976
|
Pathway
|
Known
|
Explain
|
0.03841
|
63
|
Potassium Dichromate
|
Compound
|
Known
|
Explain
|
0.03833
|
64
|
Catechin
|
Compound
|
Known
|
Explain
|
0.03802
|
65
|
ATPase activity, coupled to transmembrane movement of substances
|
Function
|
Known
|
Explain
|
0.03782
|
66
|
benzyloxycarbonylleucyl-leucyl-leucine aldehyde
|
Compound
|
Known
|
Explain
|
0.03759
|
67
|
Chromium
|
Compound
|
Known
|
Explain
|
0.03744
|
68
|
CGP 57148
|
Compound
|
Known
|
Explain
|
0.03556
|
69
|
ABCC2 gene
|
Gene
|
Inferred
|
Explain
|
0.03450
|
70
|
cellular iron ion homeostasis
|
Function
|
Known
|
Explain
|
0.03116
|
71
|
Carbamazepine
|
Compound
|
Known
|
Explain
|
0.02578
|
72
|
beta-Naphthoflavone
|
Compound
|
Known
|
Explain
|
0.02571
|
73
|
Acetaco
|
Compound
|
Known
|
Explain
|
0.02438
|
74
|
epigallocatechin gallate
|
Compound
|
Known
|
Explain
|
0.02423
|
75
|
Am 580
|
Compound
|
Known
|
Explain
|
0.02375
|
76
|
Dimethylnitrosamine
|
Compound
|
Known
|
Explain
|
0.02307
|
77
|
PD 98059
|
Compound
|
Known
|
Explain
|
0.02258
|
78
|
adenosinetriphosphatase activity
|
Function
|
Known
|
Explain
|
0.02171
|
79
|
Cadmium
|
Compound
|
Known
|
Explain
|
0.02170
|
80
|
ABC transporter-like
|
Domain
|
Known
|
Explain
|
0.02090
|
81
|
Cadmium chloride
|
Compound
|
Known
|
Explain
|
0.02078
|
82
|
zoledronic acid
|
Compound
|
Known
|
Explain
|
0.01853
|
83
|
Malignant neoplasm of breast
|
Disease
|
Known
|
Explain
|
0.01834
|
84
|
Dexamethasone
|
Compound
|
Known
|
Explain
|
0.01801
|
85
|
SMAD6 gene
|
Gene
|
Inferred
|
Explain
|
0.01773
|
86
|
Digitalis Glycosides
|
Compound
|
Inferred
|
Explain
|
0.01632
|
87
|
ATPase, AAA+ type, core
|
Domain
|
Known
|
Explain
|
0.01605
|
88
|
Cyclophosphamide
|
Compound
|
Known
|
Explain
|
0.01563
|
89
|
xenobiotic transporter activity
|
Function
|
Inferred
|
Explain
|
0.01543
|
90
|
Mitoxantrone
|
Compound
|
Known
|
Explain
|
0.01543
|
91
|
sulindac sulfide
|
Compound
|
Known
|
Explain
|
0.01522
|
92
|
Folic Acid
|
Compound
|
Known
|
Explain
|
0.01521
|
93
|
Methotrexate
|
Compound
|
Known
|
Explain
|
0.01423
|
94
|
Cardenolides
|
Compound
|
Inferred
|
Explain
|
0.01414
|
95
|
Diosmin
|
Compound
|
Inferred
|
Explain
|
0.01404
|
96
|
Topotecan
|
Compound
|
Known
|
Explain
|
0.01379
|
97
|
Mercury
|
Compound
|
Known
|
Explain
|
0.01360
|
98
|
drug response
|
Function
|
Known
|
Explain
|
0.01326
|
99
|
MVP gene
|
Gene
|
Inferred
|
Explain
|
0.01311
|
100
|
SLCO1B1 gene
|
Gene
|
Inferred
|
Explain
|
0.01288
|
|